modzatinib [Ligand Id: 14051] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| IL2 inducible T cell kinase in Human [GtoPdb: 2046] [UniProtKB: Q08881] | ||||||||
| GtoPdb | - | - | 9.74 | pIC50 | <0.18 | nM | IC50 |
WO2020033955A1. Pyrrolopyrimidine ITK inhibitors (2025); J Pharmacol Exp Ther (2025) 392: 100054 [PMID:40023606] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | - | - | 9.28 | pIC50 | <0.52 | nM | IC50 |
WO2020033955A1. Pyrrolopyrimidine ITK inhibitors (2025); J Pharmacol Exp Ther (2025) 392: 100054 [PMID:40023606] |
| TXK tyrosine kinase in Human [GtoPdb: 2268] [UniProtKB: P42681] | ||||||||
| GtoPdb | - | - | 9.08 | pIC50 | 0.83 | nM | IC50 | J Pharmacol Exp Ther (2025) 392: 100054 [PMID:40023606] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
